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| Product Name: | Catalog#: | CAS#: | Targets: | Chemical Name/IUPAC: | Chemical Formula: | Molecular Weight: |
| PLX-5622 | C-1521 | 1303420-67-8 | CSF-1R | 3-Pyridinemethanamine, 5-fluoro-N-[6-fluoro-5-[(5-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)methyl]-2-pyridinyl]-2-methoxy- | C21H19F2N5O | 395.41 |
| VG-3927 | C-1046 | - | TREM2 | - | - | - |
| Olitigaltin (TD-139, GB-0139) | C-1296 | 1450824-22-2 | Galectin-3 | (2R,2'R,3R,3'R,4S,4'S,5R,5'R,6S,6'S)-6,6'-thiobis(4-(4-(3-fluorophenyl)-1H-1,2,3-triazol-1-yl)-2-(hydroxymethyl)tetrahydro-2H-pyran-3,5-diol) | C28H30F2N6O8S | 648.64 |
| RMC-6236 | C-1418 | 2765081-21-6 | RAS(ON); RAS(MULTI)(ON) | (1S,2S)-N-((63S,4S,Z)-11-ethyl-12-(2-((S)-1-methoxyethyl)-5-(4-methylpiperazin-1-yl)pyridin-3-yl)-10,10-dimethyl-5,7-dioxo-61,62,63,64,65,66-hexahydro-11H-8-oxa-2(4,2)-thiazola-1(5,3)-indola-6(1,3)-pyridazinacycloundecaphane-4-yl)-2-methylcyclopropane-1-carboxamide | C44H58N8O5S | 811.06 |
| RMC-4630 (Vociprotafib) | C-1337 | 2172652-48-9 | SHP2 | (6-((2-amino-3-chloropyridin-4-yl)thio)-3-((3S,4S)-4-amino-3-methyl-2-oxa-8-azaspiro[4.5]decan-8-yl)-5-methylpyrazin-2-yl)methanol | C20H27ClN6O2S | 450.98 |
| RLY-4008 (Lirafugratinib) | C-1335 | 2549174-42-5 | FGFR2 | N-[4-(4-amino-5-{3-fluoro-4-[(4-methylpyrimidin-2-yl)oxy]phenyl}-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-6-yl)phenyl]-2-methylprop-2-enamide | C28H24FN7O2 | 509.53 |
